Trials / Terminated
TerminatedNCT02698176
A Dose Exploration Study With Birabresib (MK-8628) in Participants With Selected Advanced Solid Tumors (MK-8628-006)
A Phase IB Dose Exploration Trial With MK-8628, a Small Molecule Inhibitor of the Bromodomain and Extra-Terminal (BET) Proteins, in Subjects With Selected Advanced Solid Tumors
- Status
- Terminated
- Phase
- Phase 1
- Study type
- Interventional
- Enrollment
- 13 (actual)
- Sponsor
- Merck Sharp & Dohme LLC · Industry
- Sex
- All
- Age
- 18 Years
- Healthy volunteers
- Not accepted
Summary
This is a study to determine the recommended dose of birabresib (MK-8628)(formerly known as OTX015) for further studies in participants with advanced nuclear protein in testis (NUT) midline carcinoma (NMC), triple negative breast cancer (TNBC), non-small cell lung cancer (NSCLC), or castration-resistant prostate cancer (CRPC). This is a two-part parallel study: Part A will establish the recommended dose by evaluating dose limiting toxicity (DLT), safety, discontinuation, and early efficacy and Part B will enroll participants with NMC only and will evaluate safety and efficacy in this population.
Detailed description
The sponsor decided to terminate the program after evaluation of safety and efficacy data at the dose levels tested (Part A). The decision to discontinue the birabresib program was based on limited efficacy signals and was not due to safety-related concerns. No participants entered or were treated in Part B of the study.
Conditions
- NUT Midline Carcinoma (NMC)
- Triple Negative Breast Cancer (TNBC)
- Non-small Cell Lung Cancer (NSCLC)
- Castration-resistant Prostate Cancer (CRPC)
Interventions
| Type | Name | Description |
|---|---|---|
| DRUG | Birabresib | Administered as an oral capsule in a fasted state |
Timeline
- Start date
- 2016-05-04
- Primary completion
- 2017-04-26
- Completion
- 2017-04-26
- First posted
- 2016-03-03
- Last updated
- 2021-01-27
- Results posted
- 2018-11-05
Regulatory
- FDA-regulated drug study
Source: ClinicalTrials.gov record NCT02698176. Inclusion in this directory is not an endorsement.