Clinical Trials Directory

Trials / Active Not Recruiting

Active Not RecruitingNCT06462716

A Phase l Study of By101298, an Oral DNA-PK Inhibitor, in Patients With Advanced Solid Tumors

A Phase I Clinical Study to Evaluate the Safety, Tolerability, and Pharmacokinetic Characteristics of BY101298 as Single-agent Therapy/in Combination With Radiotherapy in Patients With Malignant Solid Tumors

Status
Active Not Recruiting
Phase
Phase 1
Study type
Interventional
Enrollment
36 (estimated)
Sponsor
Chengdu Baiyu Pharmaceutical Co., Ltd. · Industry
Sex
All
Age
18 Years – 75 Years
Healthy volunteers
Not accepted

Summary

BY101298 is an innovative DNA-dependent protein kinases (DNA-PK) highly selective small molecule inhibitor. DNA-dependent protein kinases (DNA-PK plays a key role in the NHEJ repair pathway to repair DNA double-strand breaks (DSBs). Primary objective is to assess the safety and tolerability of BY101298 in patients with advanced malignant solid tumors. The secondary Objectives are to characterize the pharmacokinetic (PK) profile of BY101298 in patients with advanced malignant solid tumors and to assess the preliminary efficacy of BY101298 in patients with advanced malignant solid tumors.

Conditions

Interventions

TypeNameDescription
DRUGBY101298 CapsulesAn oral DNA-PK Inhibitor

Timeline

Start date
2023-04-25
Primary completion
2024-12-31
Completion
2025-06-30
First posted
2024-06-17
Last updated
2025-04-13

Locations

1 site across 1 country: China

Source: ClinicalTrials.gov record NCT06462716. Inclusion in this directory is not an endorsement.