Trials / Recruiting
RecruitingNCT06343402
Open-label Study of BBO-8520 in Adult Subjects With KRASG12C Non-small Cell Lung Cancer
A Phase 1a/1b Open-Label Study Evaluating the Safety, Tolerability, Pharmacokinetics, and Efficacy of BBO-8520 in Subjects With Advanced KRASG12C Mutant Non-Small Cell Lung Cancer - The ONKORAS-101 Study
- Status
- Recruiting
- Phase
- Phase 1
- Study type
- Interventional
- Enrollment
- 350 (estimated)
- Sponsor
- TheRas, Inc., d/b/a BBOT (BridgeBio Oncology Therapeutics) · Industry
- Sex
- All
- Age
- 18 Years
- Healthy volunteers
- Not accepted
Summary
A first in human study to evaluate the safety and preliminary antitumor activity of BBO-8520, a KRAS G12C (ON and OFF) inhibitor, as a single agent and in combination with pembrolizumab and BBO-10203 in subjects with locally advanced and unresectable or metastatic non-small cell lung cancer with a KRAS (Kirsten rat sarcoma) G12C mutation.
Detailed description
This is an open-label, multi-center, Phase 1 study designed to evaluate the safety, tolerability, pharmacokinetics, and efficacy of BBO-8520, a direct inhibitor of KRASG12C (ON and OFF), alone and in combination with the ICI pembrolizumab and BBO-10203 in subjects with locally advanced and unresectable or metastatic non-small cell lung cancer with a KRAS (Kirsten rat sarcoma) G12C mutation. The study includes dose escalation phase and dose expansion phase
Conditions
- Non-small Cell Lung Cancer
- Metastatic Non-Small Cell Lung Cancer
- NSCLC
- KRAS G12C
- Metastatic Lung Cancer
- Advanced Lung Carcinoma
Interventions
| Type | Name | Description |
|---|---|---|
| DRUG | BBO-8520 | Participants will receive assigned dose of BBO-8520 orally (PO), QD |
| DRUG | Pembrolizumab | Patients will receive IV pembrolizumab |
| DRUG | BBO-10203 | Participants will receive assigned dose of BBO-8520 orally (PO), QD |
Timeline
- Start date
- 2024-05-22
- Primary completion
- 2031-04-01
- Completion
- 2031-09-01
- First posted
- 2024-04-02
- Last updated
- 2026-04-15
Locations
32 sites across 4 countries: United States, Australia, Canada, Spain
Regulatory
- FDA-regulated drug study
Source: ClinicalTrials.gov record NCT06343402. Inclusion in this directory is not an endorsement.