Trials / Recruiting
RecruitingNCT05902988
A Phase I/II Study of VLS-1488 in Subjects With Advanced Cancer
A Phase I/II Study of VLS-1488 (an Oral KIF18A Inhibitor) in Subjects With Advanced Cancer
- Status
- Recruiting
- Phase
- Phase 1 / Phase 2
- Study type
- Interventional
- Enrollment
- 200 (estimated)
- Sponsor
- Volastra Therapeutics, Inc. · Industry
- Sex
- All
- Age
- 18 Years
- Healthy volunteers
- Not accepted
Summary
This is a first-in-human phase I/II study to examine the safety, tolerability and preliminary efficacy of VLS-1488 in subjects with advanced cancers.
Detailed description
This a first-in-human phase I/II study designed to assess the safety, tolerability and preliminary efficacy of VLS-1488 monotherapy and consists of two parts: Dose Escalation and Dose Expansion. Dose Escalation will examine the safety and tolerability of VLS-1488 in different solid tumor types at various dose levels through a series of Dose Escalation and Backfill Cohorts to identify the Maximum Tolerated Dose (MTD) and to select dose levels for Dose Expansion. The criteria for dose (de-)escalation will be based on a Bayesian Optimal Interval (BOIN) design. Dose Expansion will examine the safety, tolerability, Drug Drug Interaction (DDI) risk, Food Effect (FE) and preliminary efficacy of VLS-1488 in different tumor types and/or dose levels of interest through various expansion cohorts. VLS-1488 will be given orally in 28-day cycles. Dosing will be continued until disease progression, unacceptable toxicity, withdrawal of consent, or other stopping criteria are met.
Conditions
- Advanced Solid Tumor
- High Grade Serous Adenocarcinoma of Ovary
- Squamous Non-small-cell Lung Cancer
- Triple Negative Breast Cancer
- Head and Neck Squamous Cell Carcinoma
- Ovarian Carcinosarcoma
- Uterine Carcinosarcoma
- Uterine Serous Carcinoma
- Endometrium Cancer
- Chromosomal Instability
Interventions
| Type | Name | Description |
|---|---|---|
| DRUG | VLS-1488 | VLS-1488 tablets will be given orally. |
Timeline
- Start date
- 2023-10-18
- Primary completion
- 2026-06-01
- Completion
- 2026-12-01
- First posted
- 2023-06-15
- Last updated
- 2025-11-04
Locations
14 sites across 1 country: United States
Regulatory
- FDA-regulated drug study
Source: ClinicalTrials.gov record NCT05902988. Inclusion in this directory is not an endorsement.