Clinical Trials Directory

Trials / Recruiting

RecruitingNCT05245500

Phase 1 Study of MRTX1719 in Solid Tumors With MTAP Deletion

A Phase 1 Multiple Expansion Cohort Trial of MRTX1719 in Patients With Advanced Solid Tumors With Homozygous MTAP Deletion

Status
Recruiting
Phase
Phase 1
Study type
Interventional
Enrollment
336 (estimated)
Sponsor
Bristol-Myers Squibb · Industry
Sex
All
Age
18 Years
Healthy volunteers
Not accepted

Summary

This is a Phase 1, open-label, multicenter, study of the safety, tolerability, PK, PD, and anti-tumor activity of MRTX1719 patients with advanced, unresectable or metastatic solid tumor malignancy with homozygous deletion of the MTAP gene.

Detailed description

This first-in-human clinical trial will begin with an exploration of MRTX1719 dose and regimen. As potentially viable regimens are identified, Phase 1b expansion cohorts may be implemented to ensure sufficient safety experience, PK information, compare food effect and relative bioavailability between capsules and tablets, and early evidence of clinical activity are available.

Conditions

Interventions

TypeNameDescription
DRUGMRTX1719MRTX1719 is a potent PRMT5-MTA inhibitor. Specified dose on specified days

Timeline

Start date
2022-06-09
Primary completion
2027-12-10
Completion
2027-12-10
First posted
2022-02-18
Last updated
2025-12-05

Locations

25 sites across 1 country: United States

Regulatory

Source: ClinicalTrials.gov record NCT05245500. Inclusion in this directory is not an endorsement.