Clinical Trials Directory

Trials / Completed

CompletedNCT05178888

Adagrasib in Combination With Palbociclib in Patients With Advanced Solid Tumors (KRYSTAL-16)

A Phase 1/1b Trial of MRTX849 in Combination With Palbociclib in Patients With Advanced Solid Tumors With KRAS G12C Mutation

Status
Completed
Phase
Phase 1
Study type
Interventional
Enrollment
11 (actual)
Sponsor
Mirati Therapeutics Inc. · Industry
Sex
All
Age
18 Years
Healthy volunteers
Not accepted

Summary

This study will evaluate the safety and clinical activity of MRTX849 (adagrasib) in combination with palbociclib in patients with advanced solid tumor malignancies with KRAS G12C mutation.

Detailed description

This study will evaluate the pharmacokinetics and preliminary clinical activity of MRTX849 (adagrasib) in combination with palbociclib in patients with advanced solid tumor malignancies with KRAS G12C mutation. MRTX849 is an orally available small molecule inhibitor of KRAS G12C and palbociclib is a small molecule inhibitor of CDK 4 and 6.

Conditions

Interventions

TypeNameDescription
DRUGMRTX849KRAS G12C inhibitor
DRUGPalbociclibCDK 4 and 6 inhibitor

Timeline

Start date
2022-01-20
Primary completion
2023-06-15
Completion
2024-12-30
First posted
2022-01-05
Last updated
2025-02-11

Locations

4 sites across 1 country: United States

Regulatory

Source: ClinicalTrials.gov record NCT05178888. Inclusion in this directory is not an endorsement.