Clinical Trials Directory

Trials / Terminated

TerminatedNCT04975256

Adagrasib in Combination With BI 1701963 in Patients With Cancer (KRYSTAL 14)

A Phase 1/1b Trial of MRTX849 in Combination With BI 1701963 in Patients With Advanced Solid Tumors With KRAS G12C Mutation

Status
Terminated
Phase
Phase 1
Study type
Interventional
Enrollment
7 (actual)
Sponsor
Mirati Therapeutics Inc. · Industry
Sex
All
Age
18 Years
Healthy volunteers
Not accepted

Summary

This study will evaluate safety, tolerability, drug levels, molecular effects and clinical activity of MRTX849 (adagrasib) in combination with BI 1701963 in patients with advanced solid tumors that have a KRAS G12C mutation.

Detailed description

This study will evaluate safety, tolerability, pharmacokinetics, metabolites, pharmacodynamics and clinical activity of MRTX849 (adagrasib) in combination with BI 1701963 in patients with advanced solid tumors with a KRAS G12C mutation. MRTX849 is an orally available small molecule inhibitor of KRAS G12C and BI 1701963 is a SOS1 pan-KRAS inhibitor.

Conditions

Interventions

TypeNameDescription
DRUGMRTX849KRAS G12C inhibitor
DRUGBI 1701963SOS1 Inhibitor

Timeline

Start date
2021-07-28
Primary completion
2022-11-02
Completion
2022-11-15
First posted
2021-07-23
Last updated
2024-12-16

Locations

4 sites across 1 country: United States

Regulatory

Source: ClinicalTrials.gov record NCT04975256. Inclusion in this directory is not an endorsement.