Clinical Trials Directory

Trials / Completed

CompletedNCT04410991

Relapsing Forms of Multiple Sclerosis (RMS) Study of Bruton's Tyrosine Kinase (BTK) Inhibitor Tolebrutinib (SAR442168) (GEMINI 2)

A Phase 3, Randomized, Double-blind Efficacy and Safety Study Comparing SAR442168 to Teriflunomide (Aubagio®) in Participants With Relapsing Forms of Multiple Sclerosis

Status
Completed
Phase
Phase 3
Study type
Interventional
Enrollment
899 (actual)
Sponsor
Sanofi · Industry
Sex
All
Age
18 Years – 55 Years
Healthy volunteers
Not accepted

Summary

Primary Objective: To assess efficacy of daily SAR442168 compared to a daily dose of 14 mg teriflunomide (Aubagio) measured by annualized adjudicated relapse rate (ARR) in participants with relapsing forms of MS Secondary Objective: To assess efficacy of SAR442168 compared to teriflunomide (Aubagio) on disability progression, MRI lesions, cognitive performance and quality of life To evaluate the safety and tolerability of daily SAR442168 To evaluate pharmacodynamics (PD) of SAR442168

Detailed description

Study duration varied per participant in this event driven trial with a treatment duration of approximately 18 to 36 months. Participants completing the study were offered to participate in a long term safety study.

Conditions

Interventions

TypeNameDescription
DRUGTolebrutinibPharmaceutical form: Tablet Route of administration: Oral
DRUGTeriflunomide HMR1726Pharmaceutical form: Tablet Route of administration: Oral
DRUGPlacebo to match TolebrutinibPharmaceutical form: Tablet Route of administration: Oral
DRUGPlacebo to match TeriflunomidePharmaceutical form: Tablet Route of administration: Oral

Timeline

Start date
2020-06-11
Primary completion
2024-07-16
Completion
2024-07-16
First posted
2020-06-01
Last updated
2025-07-02
Results posted
2025-06-18

Locations

186 sites across 28 countries: United States, Argentina, Belgium, Brazil, Canada, Chile, Croatia, Czechia, France, Germany, Greece, Hungary, India, Israel, Latvia, Netherlands, Norway, Portugal, Puerto Rico, Russia, Serbia, Slovakia, South Korea, Spain, Switzerland, Turkey (Türkiye), Ukraine, United Kingdom

Regulatory

Source: ClinicalTrials.gov record NCT04410991. Inclusion in this directory is not an endorsement.

Relapsing Forms of Multiple Sclerosis (RMS) Study of Bruton's Tyrosine Kinase (BTK) Inhibitor Tolebrutinib (SAR442168) ( (NCT04410991) · Clinical Trials Directory